Table 14: R-groups used in the design of the diversity library of AVSH analogs.
| R1 | R2 | R3 |
| 1 ...(CH2)2-Ph-(o)Cl-(p)CH3 | 1 …CH2CH(Me)(CH2)2NH2 | 1 …(CH2)2-NH2 |
| 2 ...(CH2)2-Ph-(o)NH2-(p)OH | 2 …CH2CH(Me)(CH2)2Cl | 2 …(CH2)2-O-CH3 |
| 3 ...(CH2)2-Ph-(o)Br-(p)CCl3 | 3 …CH2CH(Me)CH2NH2 | 3 …CH2-CHO |
| 4 ...(CH2)2-Ph-(o)Br-(p)OH | 4 …CH2CH(Me)2 | 4 …CH2-COCH3 |
| 5 ...(CH2)2-Ph-(o)Cl-(p)Cl | 5 …CH2CH(Me)(CH2)2OH | 5 …CH2-COCl |
| 6 ...(CH2)2-Ph-(o)F-(p)CBr3 | 6 …CH2C(Me)3 | 6 …CH2-COOCl |
| 7 ...(CH2)2-Ph-(o)F-(p)CCl3 | 7 …CH2CH(Et)2 | |
| 8 ...(CH2)2-Ph-(o)Br-(p)Cl | 8 …CH2CH(Me)C3H7 | |
| 9 ...(CH2)2-Ph-(o)Cl-(p)OH | 9 …CH2CH(Me)(CH2)2OCl | |
| 10 ...(CH2)2-Ph-(m)Cl-(p)CH3 | 10 …CH2CH(Me)C2H5 | |
| 11 ...(CH2)2-Ph-(o)NH2-(p)NO | 11 …CH2CH(Et)C3H7 | |
| 12 ...(CH2)2-Ph-(o)OH-(p)OH | ||
| 13 ...(CH2)2-Ph-(o)Br-(p)Br |